생물학적 평가
세포 기반 또는 체외 테스트에서 합성 화합물이 PPAR-바나듐 수용체를 활성화하는 능력을 테스트합니다.이 단계는 PPAR-펜타늄 활성화제로서의 잠재력을 검증하는 데 필수적입니다.
화학 원료를 구입해야하는 경우 요청 정보를 제출하여최신견적을받으십시오.
생물학적 평가의 학술 논문
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Synthesis of PPAR-γ activators inspired by the marine natural product, paecilocin A
화학 물질
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3-ethoxy-N-(p-ethoxy-phenethyl) phthalimide
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Design, synthesis, and biological evaluation of N-acetyl-2-(or 3-)carboxymethylbenzenesulfonamides as cyclooxygenase isozyme inhibitors
화학 물질
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4-fluoro-2-(methoxycarbonylmethyl)benzenesulfonamide
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Synthesis and biological evaluation of 2-epi-paclitaxel
화학 물질
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C52H73NO13Si2
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Synthesis and biological evaluation of the pyrazole class of cyclooxygenase-2-inhibitors
화학 물질
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3-(4-chlorophenyl)-1-(4-nitrophenyl)-1H-pyrazole-4-carbaldehyde
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Synthesis and biological evaluation of pyrrolidine-based T-type calcium channel inhibitors for the treatment of neuropathic pain
화학 물질
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2-(2,4-bis(trifluoromethyl)phenyl)ethanol
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Synthesis of novel structurally simplified estrogen analogues
화학 물질
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3-(2-chloro-4-hydroxyphenylethynyl)-2-methylcyclohex-2-enone
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Design, synthesis, and melatoninergic activity of new azido- and isothiocyanato-substituted indoles
화학 물질
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1H-INDOLE,3-(2-CHLOROETHYL)-5-METHOXY-
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Indole
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5- 메 톡시 인돌
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Total synthesis of the potent microtubule-stabilizing agent (+)-discodermolide
화학 물질
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2H-Pyran-2-ol, 5,6-dihydro-3,5-dimethyl-6-[(1S)-1-methyl-2-(phenylmethoxy)ethyl]-, (5S,6R)-
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Design and synthesis of thrombin receptor-derived nonpeptide mimetics utilizing a piperazine scaffold
화학 물질
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1-phenylacetyl-4-[2-(tert-butoxycarbonylamino)acetyl]piperazine
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Synthesis and biological evaluation of 3,5-disubstituted-4-alkynylisoxozales as a novel class of HSP90 inhibitors
화학 물질
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ethyl-5-(2,4-dibenzyloxy-5-isopropylphenyl)-4-iodoisoxazole-3-carboxylate
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Structural study and biological evaluation of some novel 1,2,4-triazole, thiazole, and bisthiazole derivatives bearing a sulfonamide moiety
화학 물질
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3-(6-oxo-7-phenyl-6,7-dihydro-5H-[1,2,4]triazolo-[4,3-b][1,2,4]triazol-3-yl)-N-(4-sulfamoylphenyl)propionamide
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Synthesis, biological evaluation and molecular modelling of 2,4-disubstituted-5-(6-alkylpyridin-2-yl)-1H-imidazoles as ALK5 inhibitors
화학 물질
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4-((1-hydroxy-5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methyl)benzonitrile
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TVB-2640
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SYNTHESIS OF APRAMYCIN ANALOGUES
화학 물질
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tetra-N-benzyl-5,6-O-cyclohexylidene-tetra-N-methoxycarbonylneamin
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Synthesis and biological evaluation of novel phosphoramidate derivatives of coumarin as chitin synthase inhibitors and antifungal agents
화학 물질
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phenyl(methoxyglycinyl) phosphorochloridate
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Synthesis of chiral 2-(4-phenoxyphenylsulfonylmethyl)thiiranes as selective gelatinase inhibitors
화학 물질
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(S)-2-(4-phenoxyphenylsulfanylmethyl)oxirane
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Synthesis, biological evaluation and mechanism study of a class of cyclic combretastatin A-4 analogues as novel antitumour agents
화학 물질
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2',3',4'-trimethoxyacetanilide
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1,2,3-thiadiazole thioacetanilides. Part 2: Synthesis and biological evaluation of a new series of 2-{[4-(3,4-dichlorophenyl)-1,2,3-thiadiazol-5-yl] sulfanyl}acetanilides as HIV-1 inhibitors
화학 물질
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2-{[4-(3,4-dichlorophenyl)-1,2,3-thiadiazol-5-yl]sulfanyl}-N-(2-fluorophenyl)acetamide
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Synthesis and biological evaluation of piperic acid amides as free radical scavengers and αglucosidase inhibitors
화학 물질
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(2E,4E)-5-(1,3-benzodioxol-5-yl)-N-(3-phenylpropyl)-2,4-pentadienamide
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Design, synthesis and evaluation of 3-arylidene azetidin-2-ones as potential antifungal agents against Alternaria solani Sorauer
화학 물질
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(E)-methyl 3-(4-chlorophenyl)-2-((octylamino)methyl)acrylate
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Senolytic activity of piperlongumine analogues: Synthesis and biological evaluation
화학 물질
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trans-cinnamic pivalic anhydride
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Design, synthesis, and biological evaluation of a potent, PKC selective, B-ring analog of bryostatin
화학 물질
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{(S)-3-Benzyloxy-1-[(2S,6R)-6-((R)-2,2-dimethyl-[1,3]dioxolan-4-ylmethyl)-tetrahydro-pyran-2-ylmethyl]-propoxy}-tert-butyl-diphenyl-silane
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Highly Enantioselective Synthesis of a Corey Prostaglandin Intermediate
화학 물질
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(1R,2S,4S,7R,SS)-(-)-bicyclo <2.2.1> hep-7-benzyloxymethyl-5-ene-2-p-toluenesulfinyl
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Synthesis, biological evaluation, and molecular docking studies of novel isatin-thiazole derivatives as α-glucosidase inhibitors
화학 물질
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1-METHYLISATIN, 3-THIOSEMICARBAZIDE
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Stereoselective Synthesis of an Important Prostaglandin Synthetic Intermediate
화학 물질
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(3aR,4R,5R,6aS)-5-(benzoyloxy)hexahydro-4-(iodomethyl)-2H-cyclopentafuran-2-one
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Molecular modeling of drug-pathophysiological Mtb protein targets: Synthesis of some 2-thioxo-1, 3-thiazolidin-4-one derivatives as anti-tubercular agents
화학 물질
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(Z)-5-(4-benzyloxyphenyl)methylidene-2-thioxo-4-thiazolidinone
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Total Synthesis of Antiproliferative Parvifloron F
화학 물질
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3’-isopropyl-4’,5’-dimethoxyacetophenone
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Design, synthesis, and biological evaluation of alcyopterosin a and illudalane derivatives as anticancer agents
화학 물질
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4-BroMo-5,7-diMethyl-2,3-dihydro-1H-inden-1-one
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Synthesis and Evaluation of Dolastatin 10 Analogues Containing Heteroatoms on the Amino Acid Side Chains
화학 물질
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1-Pyrrolidinecarboxylic acid, 2-[(1R,2R)-1-methoxy-2-methyl-3-oxo-3-[(2-phenylethyl)amino]propyl]-, 1,1-dimethylethyl ester, (2S)-
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Selective inhibitory activity against MAO and molecular modeling studies of 2-thiazolylhydrazone derivatives
화학 물질
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2-벤질리덴하이드라진-1-카르보티오아미드
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티오세미카르바자이드
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Design, synthesis, and biological evaluation of novel piperidine-4- carboxamide derivatives as potent CCR5 inhibitors
화학 물질
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tert-butyl 4-(4-cyanobenzylcarbamoyl)piperidine-1-carboxylate
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Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin- 2-yl)-4-(quinolin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors
화학 물질
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2-(3-(6-methylpyridin-2-yl)-4-(quinolin-6-yl)-1H-pyrazol-1-yl)-N-phenylacetamide
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5-HT6 receptor antagonists: lead optimisation and biological evaluation of N-aryl and N-heteroaryl 4-amino-benzene sulfonamides
화학 물질
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N-[4-(6-chloro-2-isopropylamino-pyrimidin-4-ylsulfamoyl)-phenyl]-acetamide
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Synthesis and biological evaluation of 4-(pyridin-4-oxy)-3-(3,3-difluorocyclobutyl)-pyrazole derivatives as novel potent transforming growth factor-β type 1 receptor inhibitors
화학 물질
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2-bromo-1-(3,3-difluorocyclobutyl)ethan-1-one
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Total Synthesis of Halicholactone and Neohalicholactone
화학 물질
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2(3H)-Furanone, dihydro-4-[(4-methoxyphenyl)methoxy]-, (4S)-
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Design, synthesis and biological evaluation of novel thieno[3,2-d] pyrimidine derivatives containing diaryl urea moiety as potent antitumor agents
화학 물질
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2-(4-nitrophenyl)-4-hydroxythieno[3,2-d]pyrimidine
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Synthesis and biological evaluation of quinazoline derivatives – A SAR study of novel inhibitors of ABCG2
화학 물질
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4-phenoxy-2-phenylquinazoline
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Synthesis and biological evaluation of a focused library of beauveriolides
화학 물질
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C27H43N3O6*ClH
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Design and synthesis of triarylacrylonitrile analogues of tamoxifen with improved binding selectivity to protein kinase C
화학 물질
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Benzeneacetonitrile, a-[bis[4-[2-(diethylamino)ethoxy]phenyl]methylene]-
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Lead structures for applications in photodynamic therapy. Part 1: Synthesis and variation of m-THPC (Temoporfin) related amphiphilic A2BC-type porphyrins
화학 물질
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5,10,15,20-tetra(n-hexyl)phorphyrin
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